期刊文献

Therapeutic Potential of Lythrum salicaria L. Ethanol Extract in Experimental Rat Models of Streptozotocin-Induced Diabetes Mellitus and Letrozole-Induced Polycystic Ovary Syndrome 收藏

链霉菌素诱导的糖尿病和letrozole诱导的多囊卵巢综合征的实验大鼠模型中溶血性盐乳杆菌提取物的治疗潜力
摘要
Polycystic ovary syndrome (PCOS) and diabetes mellitus (DM) are prevalent endocrine disorders with overlapping pathophysiological mechanisms. Type 2 diabetes mellitus (T2DM) is commonly associated with PCOS, with both conditions strongly linked to insulin resistance (IR), while recent studies have also reported an increased prevalence of PCOS among women with type 1 diabetes mellitus (T1DM). This study evaluated the potential of Lythrum salicaria L. ethanol extract (LSEE) to mitigate oxidative stress (OS), inflammation, and metabolic and hormonal imbalances in separate experimental models of Streptozotocin (STZ)-induced DM and Letrozole (LET)-induced PCOS. LSEE underwent phytochemical analysis to quantify total phenolic and flavonoid content and HPLC-MS for polyphenols identification. In vitro, antioxidant capacity was investigated through FRAP, DPPH, NO, and H2O2 scavenging assays. Subsequently, in vivo, studies utilized STZ-induced DM and LET-induced PCOS rat models, with 10-day treatments of LSEE, metformin, or trolox (TX) administered by gavage. Dysregulation of hormonal profiles, ultrasound, and histological examinations confirmed PCOS development. At the end of the treatment period, serum samples were collected to assess OS markers (TOS, OSI, MDA, AOPP, 8-OHdG, NO, 3-NT, AGEs, TAR, SH) in both models. Inflammatory markers were also measured (IL-1β, NF-κB, IL-18, and Gasdermin D in DM and IL-1β, NF-κB, IL-18, and IL-10 in PCOS). Additionally, metabolic markers (glucose, lipids, TG-glucose index, liver enzymes) were assessed in DM rats, and hormones (LH, FSH, estrogen, testosterone, insulin, HOMA-IR) were determined in PCOS rats. LSEE demonstrated a high polyphenolic content and notable in vitro antioxidant activity. In vivo, it effectively reduced OS by lowering oxidant levels and enhancing antioxidant defenses, reduced inflammatory markers and blood glucose levels, and improved lipid profiles along with the TyG index and liver injury markers in diabetic rats. In PCOS rats, LSEE lowered the total oxidants, increased antioxidants, reduced LH, FSH, testosterone, and insulin, and increased estrogen levels. The effects exhibited a dose-dependent pattern, with higher doses producing more pronounced benefits comparable to those observed with metformin and TX. In conclusion, LSEE may be a promising complementary treatment for DM and PCOS.
摘要译文
多囊卵巢综合征(PCOS)和糖尿病(DM)是具有重叠的病理生理机制的普遍内分泌疾病。2型糖尿病(T2DM)通常与PCOS相关,这两种疾病都与胰岛素抵抗(IR)密切相关,而最近的研究也报道了1型1型糖尿病女性PCOS的患病率增加了。这项研究评估了在单独的链链球菌素(STZ)诱导的DM和LeTrozole(LeTrozole(LeTrozole)(LET)诱导的PCOS的实验模型中,评估了减轻氧化应激(OS),炎症以及代谢和激素失衡的潜力。LSEE进行了植物化学分析,以量化多酚鉴定的总酚类和类黄酮含量以及HPLC-MS。在体外,通过FRAP,DPPH,NO和H2O2清除测定法研究了抗氧化能力。随后,在体内,研究利用了STZ诱导的DM和Let-ty-PCOS大鼠模型,并使用了10天的LSEE,二甲双胍或Trolox(TX)治疗,该治疗方法是通过Gavage施用的。激素特征,超声检查和组织学检查的失调证实了PCOS的发展。在治疗期结束时,收集血清样品以评估OS标记(TOS,OSI,MDA,AOPP,8-OHDG,NO,3-NT,AGES,AGES,TAR,SH)。还测量了炎症标志物(在DM和IL-1β,NF-κB,NF-κB,IL-18和IL-10中,IL-1β,NF-κB,IL-18和Gasdermin D中的PCOS中)。另外,在DM大鼠中评估了代谢标记(葡萄糖,脂质,TG-葡萄糖指数,肝酶),在PCOS大鼠中测定了激素(LH,FSH,FSH,雌激素,睾丸激素,胰岛素,HOMA-IR)。LSEE表现出高的多酚含量和值得注意的体外抗氧化活性。在体内,它通过降低氧化剂水平并增强抗氧化剂防御能力,降低炎症标记和血糖水平以及改善脂质谱以及糖尿病大鼠的TYG指数和肝损伤标记,从而有效地降低了OS。在PCOS大鼠中,LSEE降低了总氧化剂,抗氧化剂增加,LH,FSH,睾丸激素和胰岛素减少,雌激素水平升高。该作用表现出剂量依赖性的模式,较高剂量产生的益处与二甲双胍和TX观察到的益处相当。总之,LSEE可能是DM和PCOS的有前途的互补疗法。
Lia Oxana Usatiuc; Marcel Pârvu; Raluca Maria Pop; Ana Uifălean; Dan Vălean; Adrian Surd; Mădălina Țicolea; Ana Hîruța; Floricuța Ranga; Florinela Adriana Cătoi; Corina Cătană; Alina Elena Pârvu. Therapeutic Potential of Lythrum salicaria L. Ethanol Extract in Experimental Rat Models of Streptozotocin-Induced Diabetes Mellitus and Letrozole-Induced Polycystic Ovary Syndrome[J]. Antioxidants, 2025,14(5): 573